上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白,专注于信号通路和疾病研究领域。
DP-C-4 纯度: 99.72%
DP-C-4 是一种基于 Cereblon 的双 PROTAC,用于同时降解 EGFR 和 PARP。
DP-C-4 Chemical Structure
规格 | 价格 | 是否有货 | 数量 |
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1 mg | ¥2800 | In-stock | |
5 mg | ¥8500 | In-stock | |
10 mg | ¥13500 | In-stock | |
50 mg | 询价 | ||
100 mg | 询价 |
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DP-C-4 相关产品
•相关化合物库:
- Bioactive Compound Library Plus
生物活性 |
DP-C-4 is a Cereblon-based dual PROTAC for simultaneous degradation of EGFR and PARP[1]. |
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IC50 & Target[1] |
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体外研究 (In Vitro) |
DP-C-4 (1-50 μM; 24 hours) has degradation effects on EGFR and PARP simultaneously in a dose-dependent manner in SW1990 cells[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. Western Blot Analysis[1]
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分子量 |
1450.93 |
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Formula |
C72H78ClF2N15O14 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
-80°C, stored under nitrogen |
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溶解性数据 |
In Vitro:
DMSO : 12 mg/mL (8.27 mM; Need ultrasonic) 配制储备液
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请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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