上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。
DDR1-IN-5
DDR1-IN-5 是选择性的盘状结构域受体家族成员 1 (DDR1) 抑制剂，IC50 为 7.36 nM。DDR1-IN-5 抑制 DDR1b (Y513) 自磷酸化，IC50 为 4.1 nM。DDR1-IN-5 具有抗癌活性。
DDR1-IN-5 Chemical Structure
CAS No. : 2416022-90-5
| 规格 | 是否有货 | ||
|---|---|---|---|
| 100 mg | 询价 | ||
| 250 mg | 询价 | ||
| 500 mg | 询价 |
* Please select Quantity before adding items.
| 生物活性 |
DDR1-IN-5 is a selective Discoidin Domain Receptor family, member 1 (DDR1) inhibitor with an IC50 of 7.36 nM. DDR1-IN-5 inhibits auto-phosphorylation DDR1b (Y513) with an IC50 of 4.1 nM. DDR1-IN-5 has anti-cancer activity[1]. |
|
|---|---|---|
| IC50 & Target[1] |
|
|
| 体外研究 (In Vitro) |
DDR1-IN-5 (compound 121; for 24 hours) inhibits collagen production in human hepatic stellate cell LX-2 (IC50=62 nM)[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
|
| 分子量 |
434.37 |
|
| Formula |
C22H13F3N6O |
|
| CAS 号 |
2416022-90-5 |
|
| 运输条件 |
Room temperature in continental US; may vary elsewhere. |
|
| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis. |
|
| 参考文献 |
|
所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务