标签归档：par

PAR-2-IN-1

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上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

PAR-2-IN-1  纯度: 99.16%

PAR-2-IN-1 是一种蛋白酶激活的受体 2 (PAR2) 信号通路抑制剂，具有抗炎和抗癌作用。

PAR-2-IN-1

PAR-2-IN-1 Chemical Structure

CAS No. : 1690176-75-0

规格 价格 是否有货 数量
Free Sample (0.1-0.5 mg)   Apply now  
5 mg ￥1000 In-stock
10 mg ￥1700 In-stock
25 mg ￥3500 In-stock
50 mg ￥5500 In-stock
100 mg ￥9500 In-stock
200 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

PAR-2-IN-1 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • GPCR/G Protein Compound Library
  • Immunology/Inflammation Compound Library
  • Anti-Cancer Compound Library

生物活性

PAR-2-IN-1 is a protease-activated receptor-2 (PAR2) signaling pathway inhibitor with anti-inflammatory and anticancer effects[1].

IC50 & Target

PAR2[1]
分子量

267.71

Formula

C12H14ClN3O2
CAS 号

1690176-75-0
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
In solvent -80°C 6 months
-20°C 1 month
溶解性数据
In Vitro: 

DMSO : 83.33 mg/mL (311.27 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 3.7354 mL 18.6769 mL 37.3539 mL
5 mM 0.7471 mL 3.7354 mL 7.4708 mL
10 mM 0.3735 mL 1.8677 mL 3.7354 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。

In Vivo:

请根据您的实验动物和给药方式选择适当的溶解方案。以下溶解方案都请先按照 In Vitro 方式配制澄清的储备液，再依次添加助溶剂：

——为保证实验结果的可靠性，澄清的储备液可以根据储存条件，适当保存；体内实验的工作液，建议您现用现配，当天使用； 以下溶剂前显示的百
分比是指该溶剂在您配制终溶液中的体积占比；如在配制过程中出现沉淀、析出现象，可以通过加热和/或超声的方式助溶

  • 1.

    请依序添加每种溶剂： 10% DMSO    90% corn oil

    Solubility: ≥ 2.08 mg/mL (7.77 mM); Clear solution

    此方案可获得 ≥ 2.08 mg/mL (7.77 mM，饱和度未知) 的澄清溶液，此方案不适用于实验周期在半个月以上的实验。

    以 1 mL 工作液为例，取 100 μL 20.8 mg/mL 的澄清 DMSO 储备液加到 900 μL玉米油中，混合均匀。

*以上所有助溶剂都可在 上海金畔生物科技有限公司 网站选购。
参考文献

  • [1]. Luc J. Farmer, et al. Imidazopyridazines useful as inhibitors of the par-2 signaling pathway. WO2015048245A1.

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Protease-Activated Receptor-1, PAR-1 Agonist TFA

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

Protease-Activated Receptor-1, PAR-1 Agonist TFA  纯度: 99.08%

Protease-Activated Receptor-1, PAR-1 Agonist TFA 是一种选择性蛋白酶激活受体1 (PAR-1) 激动肽。Protease-Activated Receptor-1, PAR-1 Agonist TFA 对应于 PAR1 配体，可通过该受体选择性地模拟凝血酶的作用。

Protease-Activated Receptor-1, PAR-1 Agonist TFA

Protease-Activated Receptor-1, PAR-1 Agonist TFA Chemical Structure

规格 价格 是否有货 数量
10 mg ￥4250 In-stock
50 mg   询价  
100 mg   询价  

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Protease-Activated Receptor-1, PAR-1 Agonist TFA 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • GPCR/G Protein Compound Library
  • Immunology/Inflammation Compound Library
  • Anti-Cancer Compound Library
  • Peptide Library

生物活性

Protease-Activated Receptor-1, PAR-1 Agonist TFA is a selective proteinase-activated receptor1 (PAR-1) agonist peptide. Protease-Activated Receptor-1, PAR-1 Agonist TFA corresponds to PAR1 tethered ligand and which can selectively mimic theactions of thrombin via this receptor[1][2].

体外研究
(In Vitro)

Protease-Activated Receptor-1, PAR-1 Agonist induces activation of protein kinase C isoenzymes alpha and epsilon in human HT-29 colon carcinoma cells expressing PAR1 endogeneously. On the cellular level, Protease-Activated Receptor-1, PAR-1 Agonist and thrombin prompted HT-29 cell migration and matrix adhesion by a PKCepsilon-dependent mechanism as concluded because of the inhibition of PAR1-mediated effects by the PKC inhibitor bisindolylmaleimide I and the PKCepsilon translocation inhibitory peptide EAVSLKPT but not by the PKC inhibitor Gö 6976[2].

上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

876.92

Formula

C37H59F3N10O11
Sequence

Thr-Phe-Leu-Leu-Arg-Asn
Sequence Shortening

TFLLRN
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Sealed storage, away from moisture

Powder -80°C 2 years
-20°C 1 year

*In solvent : -80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)
溶解性数据
In Vitro: 

H2O : 6.67 mg/mL (7.61 mM; ultrasonic and warming and heat to 60°C)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 1.1404 mL 5.7018 mL 11.4035 mL
5 mM 0.2281 mL 1.1404 mL 2.2807 mL
10 mM — — —

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month (sealed storage, away from moisture)。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Stefanie Gödecke, et al. Thrombin-induced ATP release from human umbilical vein endothelial cells. Am J Physiol Cell Physiol. 2012 Mar 15;302(6):C915-23.

    [2]. Heider I, et al. PAR1-type thrombin receptor stimulates migration and matrix adhesion of human colon carcinoma cells by a PKCepsilon-dependent mechanism. Oncol Res. 2004;14(10):475-482.

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多肽定制PAR – 1 Agonist;Protease – Activated Recep,Protease Activated Receptor-1-selective peptide 编码

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名称 PAR – 1 Agonist;Protease – Activated Recep,Protease Activated Receptor-1-selective peptide
编码
别名 PAR – 1 Agonist;Protease – Activated Recep,Protease Activated Receptor-1-selective peptide
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） TFLLRN
序列（三字母缩写） H-Thr-Phe-Leu-Leu-Arg-Asn-OH (trifluoroacetate salt)
基本描述 PAR1 Agonist.
溶解度
分子量 762.9
化学式 C35H58N10O9
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR - 1 Agonist;Protease - Activated Recep,Protease Activated Receptor-1-selective peptide 编码
Figures PAR - 1 Agonist;Protease - Activated Recep,Protease Activated Receptor-1-selective peptide 编码
Reference Syeda,, F. et al. J. Biol. Chem 281, 11792 (2006) Jenkins, R. et al. J. Clin. Invest 116, 1606 (2006)
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多肽定制PAR-1,Protease Activated Receptor-1(1-6)) (mouse, rat) 编码 [140436-67-5]

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上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-1,Protease Activated Receptor-1(1-6)) (mouse, rat)
编码 [140436-67-5]
别名 PAR-1,Protease Activated Receptor-1(1-6)) (mouse, rat)
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） SFFLRN
序列（三字母缩写） H-Ser-Phe-Phe-Leu-Arg-Asn-OH (trifluoroacetate salt)
基本描述 This peptide inhibited activation of PAR-2 by trypsin in PAR-2 receptor expressing KNRK cells. Half-maximal inhibition of calcium signaling was observed at about 50 碌M. In contrast, the activation of PAR-2 by SLIGRL-NH2 (PAR-2 (1-6) amide (mouse, rat)) was not inhibited by this peptide. Selective Antagonist for PAR2 Agonist. This peptide blocks trypsin but not SLIGRL-NH2 activation of PAR2 in receptor-expressing KNRK cells.
溶解度
分子量 782.9
化学式 C37H54N10O9
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-1,Protease Activated Receptor-1(1-6)) (mouse, rat) 编码 [140436-67-5]
Figures PAR-1,Protease Activated Receptor-1(1-6)) (mouse, rat) 编码 [140436-67-5]
Reference Z.Suo et al., J. Biol. Chem., 278, 37681 (2003) P.J.Yu et al., Oncogene, 27, 2594 (2008) F.Bock et al., Proc. Natl. Acad. Sci. USA, 110, 648 (2013)
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多肽定制PAR-2 (1-6)) amide (human)) (scrambled) 编码

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上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-2 (1-6)) amide (human)) (scrambled)
编码
别名 PAR-2 (1-6)) amide (human)) (scrambled)
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） LSIGKV-NH2
序列（三字母缩写） H-Leu-Ser-Ile-Gly-Lys-Val-NH2?(trifluoroacetate salt)
基本描述 The peptide T1 is the thrombin receptor domain, which functions as a tethered ligand for the receptor itself. T1 is an inhibitor of thrombin triggered platelet aggregation, serotonin release and tyrosine phosphorylation. Its anti-aggregatory activity was about ten-fold higher than that of the previously reported peptide antagonists of the thrombin receptor. This peptide has served as model peptide in protein modification and MS studies.
溶解度
分子量 614.79
化学式 C28H54N8O7
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-2 (1-6)) amide (human)) (scrambled) 编码
Figures PAR-2 (1-6)) amide (human)) (scrambled) 编码
Reference H.Nishikawa et al., J. Pharmacol. Exp. Ther., 312, 324 (2005) I.A. Akers et al.,Am. J. Physiol. Lung Cell. Mol. Physiol., 278, L193 (2000) S. Miyata, et al., J. Biol. Chem., 275, 4592 (2000) S. Miike, A.S. McWilliam, and H. Kita, J. Immunol., 167, 6615 (2001)
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多肽定制PAR-2 (1-6),Protease Activated Receptor-2 (1-6), (mouse, rat) 编码 [164081-25-8]

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上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-2 (1-6),Protease Activated Receptor-2 (1-6), (mouse, rat)
编码 [164081-25-8]
别名 PAR-2 (1-6),Protease Activated Receptor-2 (1-6), (mouse, rat)
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） SLIGRL
序列（三字母缩写） H-Ser-Leu-Ile-Gly-Arg-Leu-OH (trifluoroacetate salt)
基本描述 The peptide is a protease-activated receptor-2 (PAR2) selective agonist.
溶解度
分子量 657.81
化学式 C29H55N9O8
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-2 (1-6),Protease Activated Receptor-2 (1-6), (mouse, rat) 编码 [164081-25-8]
Figures PAR-2 (1-6),Protease Activated Receptor-2 (1-6), (mouse, rat) 编码 [164081-25-8]
Reference R.J.Santulli et al., Proc. Natl. Acad. Sci. USA, 92, 9151 (1995) A. Bhattacharya et al., J. Pharmacol. Exp. Ther., 297, 573 (2001) B. Al-Ani, et al., J. of Physiol. Pharmacol., 73, 1203 (1995)
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多肽定制PAR-2 (1-6),Protease Activated Receptor-2 (1-6),amide (mouse, rat) 编码 [171436-38-7]

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上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-2 (1-6),Protease Activated Receptor-2 (1-6),amide (mouse, rat)
编码 [171436-38-7]
别名 PAR-2 (1-6),Protease Activated Receptor-2 (1-6),amide (mouse, rat)
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） SLIGRL-NH2
序列（三字母缩写） H-Ser-Leu-Ile-Gly-Arg-Leu-NH2?(trifluoroacetate salt)
基本描述 This peptide mimicks the putative tethered ligand of human PAR-3 (protease activated receptor 3). PAR3 Tethered Ligand (Human) / Activates PAR1 and PAR2
溶解度
分子量 656.83
化学式 C29H56N10O7
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-2 (1-6),Protease Activated Receptor-2 (1-6),amide (mouse, rat) 编码 [171436-38-7]
Figures PAR-2 (1-6),Protease Activated Receptor-2 (1-6),amide (mouse, rat) 编码 [171436-38-7]
Reference B.al-Ani et al., Can. J. Physiol. Pharmacol., 73, 1203 (1995) M.D.Hollenberg et al., Mol. Pharmacol., 49, 229 (1996) M.Saiffeddine et al., Br. J. Pharmacol., 118, 521 (1996) N.Vergnolle, J. Immunol., 163, 5064 (1999) B.Al-Ani et al., Br. J. Pharmacol., 128, 1105 (1999) E.R.Sharlow et al., J. Cell Sci., 113, 3093 (2000)
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多肽定制PAR-3 (1-6),Protease Activated Receptor-3 (1-6), human 编码 [320347-28-2]

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上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-3 (1-6),Protease Activated Receptor-3 (1-6), human
编码 [320347-28-2]
别名 PAR-3 (1-6),Protease Activated Receptor-3 (1-6), human
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） TFRGAP
序列（三字母缩写） H-Thr-Phe-Arg-Gly-Ala-Pro-OH (trifluoroacetate salt)
基本描述 This peptide is a human PAR-3-derived tethered ligand, which does not activate PAR-3 but rather activates PAR-1 and PAR-2, either in Jurkat or in other PAR-expressing cells. PAR3 Tethered Ligand (Human) / Activates PAR1 and PAR2 This peptide is the 1-6 fragment of the protease-activated receptor 3 (PAR-3), which induces ERK activation in human carcinoma cells endogeneously expressing PAR1 and PAR3. This effect is completely abolished by single alanine substitution at positions 3, 4 and 6 in the peptide. PAR-3 allosterically regulates PAR1 signaling by receptor dimerization governing increased endothelial permeability. Targeting of PAR3 may mitigate the effects of PAR1 in activating endothelial responses such as vascular inflammation. However this peptide does not affect VEGF release or expression.
溶解度
分子量 647.73
化学式 C29H45N9O8
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-3 (1-6),Protease Activated Receptor-3 (1-6), human 编码 [320347-28-2]
Figures PAR-3 (1-6),Protease Activated Receptor-3 (1-6), human 编码 [320347-28-2]
Reference H.Ishihara et al., Nature, 386, 502 (1997) K.K. Hansen et al., Immunology, 112, 183 (2004)
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多肽定制PAR-3 (1-6)Protease Activated Receptor-3 (1-6) amide, human 编码

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-3 (1-6)Protease Activated Receptor-3 (1-6) amide, human
编码
别名 PAR-3 (1-6)Protease Activated Receptor-3 (1-6) amide, human
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） TFRGAP-NH2
序列（三字母缩写） H-Thr-Phe-Arg-Gly-Ala-Pro-NH2?(trifluoroacetate salt)
基本描述 This peptide is a murine PAR-3-derived tethered ligand sequence which does not activate PAR-3, but rather activates PAR-1 and PAR-2, either in Jurkat T-cells or in other PAR-expressing cells. PAR3 Tethered Ligand (Murine) / Activates PAR1 and PAR2
溶解度
分子量 646.75
化学式 C29H46N10O7
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-3 (1-6)Protease Activated Receptor-3 (1-6) amide, human 编码
Figures PAR-3 (1-6)Protease Activated Receptor-3 (1-6) amide, human 编码
Reference K.K.Hansen et al., Immunology, 112, 183 (2004) Kaufmann, R. et al. Regul. Pept. 125, 61( 2005) McLaughlin, J. et al. PNAS 104, 5662 (2007) Arisato, T. et al. Cell. Mol. Life Sci. 60, 1420 (2003)
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多肽定制PAR-3 ,Protease Activated Receptor-3(1-6)) amide (mouse) 编码 [261521-21-5]

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-3 ,Protease Activated Receptor-3(1-6)) amide (mouse)
编码 [261521-21-5]
别名 PAR-3 ,Protease Activated Receptor-3(1-6)) amide (mouse)
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） SFNGGP-NH2
序列（三字母缩写） H-Ser-Phe-Asn-Gly-Gly-Pro-NH2?(trifluoroacetate salt)
基本描述 This peptide is the amino terminus of the fourth protease-activated receptor (PAR4) after the cleavage at Arg47/Gly48 was tested for its ability to stimulate COS cells expressing PAR4. The peptide readily activated both wild-type and mutant PAR4 (R47A) at 500 碌M, whereas thrombin and trypsin only activate the wild-type PAR4.
溶解度
分子量 576.61
化学式 C25H36N8O8
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-3 ,Protease Activated Receptor-3(1-6)) amide (mouse) 编码 [261521-21-5]
Figures PAR-3 ,Protease Activated Receptor-3(1-6)) amide (mouse) 编码 [261521-21-5]
Reference K.K.Hansen et al., Immunology, 112, 183 (2004)
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多肽定制PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, human 编码 [245443-51-0]

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, human
编码 [245443-51-0]
别名 PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, human
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） GYPGQV-NH2
序列（三字母缩写） H-Gly-Tyr-Pro-Gly-Gln-Val-NH2
基本描述 Protease-activated receptor-4 activating peptide derived from murine PAR-4. This peptide was able to cause rat platelet aggregation with an EC50 value of 40 碌M. Its effect on leucocyte rolling and adherence points at a role of PAR-4 in mediating proinflammatory processes. The family of at least seven transmembrane G protein coupled receptors includes at least four receptor subtypes (PAR1, PAR2, PAR3, PAR4). PAR4 activating peptides, GYPGKF-NH2 and AYPGKG-NH2, produce concentration dependent contractile effects on the muscle.
溶解度
分子量 618.69
化学式 C28H42N8O8
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, human 编码 [245443-51-0]
Figures PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, human 编码 [245443-51-0]
Reference M.D.Hollenberg et al., Can. J. Physiol. Pharmacol., 77, 458 (1999) M.Tognetto et al., Br. J. Pharmacol., 139, 21 (2003) M.D.Hollenberg and S.Houle, Swiss Med. Wkly., 135, 425 (2005)
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多肽定制PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, mouse 编码 [245443-52-1]

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, mouse
编码 [245443-52-1]
别名 PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, mouse
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） GYPGKF-NH2
序列（三字母缩写） H-Gly-Tyr-Pro-Gly-Lys-Phe-NH2?(trifluoroacetate salt)
基本描述 This peptide based on the proteolytically-revealed tethered ligand sequence of the murine proteinase-activated receptor-4 (PAR-4) was shown to cause platelet aggregation with an EC50 value of about 15 碌M. PAR-4 agonist peptide stimulates thromboxane production by human platelets with the maximal response to this agonist being approximately half of that observed after maximal thrombin stimulation.
溶解度
分子量 666.78
化学式 C33H46N8O7
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, mouse 编码 [245443-52-1]
Figures PAR-4 (1-6)) amide |Protease Activated Receptor-4 (1-6) amide, mouse 编码 [245443-52-1]
Reference N.Vergnolle, J. Immunol., 163, 5064 (1999) M.D.Hollenberg and M.Saifeddine, Can. J. Physiol. Pharmacol., 79, 439 (2001) Fang, J. et al. Blood 106, 2671(2005) Mulè, F. et al. Gut. 53, 229 (2004) Sekiguchi, F. et al. Drug Design Rev. 1, 287 (2004) Faruqi, T. et al. J. Biol. Chem. 275, 19728 (2000) Greenberg, D. Biochem. 42, 2702 (2003)
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多肽定制PAR-4 (1-6)) |Protease Activated Receptor-4 (1-6), human 编码 [225779-44-2]

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-4 (1-6)) |Protease Activated Receptor-4 (1-6), human
编码 [225779-44-2]
别名 PAR-4 (1-6)) |Protease Activated Receptor-4 (1-6), human
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） GYPGQV
序列（三字母缩写） H-Gly-Tyr-Pro-Gly-Gln-Val-OH (trifluoroacetate salt)
基本描述 This PAR-4 activating peptide caused secretion and aggregation of PAR-3 deficient mouse platelets.
溶解度
分子量 619.68
化学式 C28H41N7O9
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-4 (1-6)) |Protease Activated Receptor-4 (1-6), human 编码 [225779-44-2]
Figures PAR-4 (1-6)) |Protease Activated Receptor-4 (1-6), human 编码 [225779-44-2]
Reference W.-F.Xu et al., Proc. Natl. Acad. Sci. USA, 95, 6642 (1998) H.Andersen et al., Proc. Natl. Acad. Sci. USA, 96, 11189 (1999) R.Kaufmann et al., J. Cancer Res. Clin. Oncol., 126, 91 (2000)
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多肽定制PAR-4 (1-6))|Protease Activated Receptor-4 (1-6), mouse 编码 [213018-42-9]

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-4 (1-6))|Protease Activated Receptor-4 (1-6), mouse
编码 [213018-42-9]
别名 PAR-4 (1-6))|Protease Activated Receptor-4 (1-6), mouse
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） GYPGKF
序列（三字母缩写） H-Gly-Tyr-Pro-Gly-Lys-Phe-OH (trifluoroacetate salt)
基本描述
溶解度
分子量 667.76
化学式 C33H45N7O8
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-4 (1-6))|Protease Activated Receptor-4 (1-6), mouse 编码 [213018-42-9]
Figures PAR-4 (1-6))|Protease Activated Receptor-4 (1-6), mouse 编码 [213018-42-9]
Reference M.L.Kahn et al., Nature, 394, 690 (1998)
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多肽定制PAR-2 Agonis,Protease-Activated Receptor-2 Agonist amide 编码

发表于由

上海金畔生物科技有限公司可以定制不同序列多肽，可以访问官网了解更多产品信息。

名称 PAR-2 Agonis,Protease-Activated Receptor-2 Agonist amide
编码
别名 PAR-2 Agonis,Protease-Activated Receptor-2 Agonist amide
纯度 80%，90%，95%，98%，99%
重量 1mg,5mg,10mg,50mg,100mg,1g
序列（单字母缩写） SLIGKV-NH2
序列（三字母缩写） H-Ser-Leu-Ile-Gly-Lys-Val-NH2?(trifluoroacetate salt)
基本描述
溶解度
分子量 614.8
化学式 C28H54N8O7
存储条件 Store at -20°C. Keep tightly closed. Store in a cool dry place.
注释
Documents PAR-2 Agonis,Protease-Activated Receptor-2 Agonist amide 编码
Figures PAR-2 Agonis,Protease-Activated Receptor-2 Agonist amide 编码
Reference Dulon et al. Am. J. Resp. Cell Mol. Biol. 28, 339 (2003) Kim, M. et al. Cell Biochem. Funct. 20, 339 (2002) Vesey, D. et al. Kidney International 67, 1315 (2005) Hollenberg, M. Can. J. Physiol. Pharmacol. 75, 832 (1997) Nishikawa, H. et al. J. Pharmacol. Exp. Ther. 312, 324 (2005)
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