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EMI48 纯度: 99.02%
EMI48 是 EMI1 的衍生物,EMI48 比 EMI1 对突变型 EGFR 具有更大的效力。EMI48 抑制 EGFR 三重突变体。
EMI48 Chemical Structure
CAS No. : 34564-13-1
规格 | 价格 | 是否有货 | 数量 |
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10 mM * 1 mL in DMSO | ¥3300 | In-stock | |
5 mg | ¥3000 | In-stock | |
10 mg | ¥4800 | In-stock | |
50 mg | ¥14000 | In-stock | |
100 mg | ¥20000 | In-stock | |
200 mg | 询价 | ||
500 mg | 询价 |
* Please select Quantity before adding items.
EMI48 相关产品
•相关化合物库:
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生物活性 |
EMI48, the derivative of EMI1, displays greater potency toward mutant EGFR than EMI1. EMI48 inhibits EGFR triple mutants[1]. |
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IC50 & Target[1] |
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体外研究 (In Vitro) |
EMI48 inhibits EGFR ex19del/T790M/C797S and EGFR L858R/T790M/C797S. EMI48 can be used in the research of mutant EGFR-associated, drug-resistant non-small-cell lung cancer (NSCLC)[1]. Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only. |
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分子量 |
348.40 |
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Formula |
C21H20N2O3 |
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CAS 号 |
34564-13-1 |
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运输条件 |
Room temperature in continental US; may vary elsewhere. |
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储存方式 |
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溶解性数据 |
In Vitro:
DMSO : 9.26 mg/mL (26.58 mM; Need ultrasonic) 配制储备液
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请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液;一旦配成溶液,请分装保存,避免反复冻融造成的产品失效。 |
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参考文献 |
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