PGAM1-IN-1

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PGAM1-IN-1  纯度: 99.35%

PGAM1-IN-1 是一种有效的磷酸甘油酸变位酶 1 (PGAM1) 抑制剂，IC50 为 6.4 μM。

PGAM1-IN-1

PGAM1-IN-1 Chemical Structure

CAS No. : 2438637-65-9

规格 价格 是否有货 数量
10 mM * 1 mL in DMSO ￥3850 In-stock
5 mg ￥3500 In-stock
10 mg ￥5500 In-stock
50 mg ￥16500 In-stock
100 mg   询价  
200 mg   询价  

* Please select Quantity before adding items.

PGAM1-IN-1 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Metabolism/Protease Compound Library
  • Anti-Cancer Compound Library
  • Glycolysis Compound Library
  • Phosphatase Inhibitor Library
  • Anti-Cancer Metabolism Compound Library
  • Glucose Metabolism Compound Library

生物活性

PGAM1-IN-1 is a phosphoglycerate mutase 1 (PGAM1) inhibitor with an IC50 of 6.4 μM[1].

IC50 & Target

IC50: 6.4 μM (PGAM1)[1]
体外研究
(In Vitro)

PGAM1-IN-1 (Compound 9h) inhibits H1299 proliferation with an IC50 of 14.1±1.9 μM[1].

上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

435.81

Formula

C19H11ClFNO6S
CAS 号

2438637-65-9
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
溶解性数据
In Vitro: 

DMSO : 5 mg/mL (11.47 mM; Need ultrasonic and warming)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 2.2946 mL 11.4729 mL 22.9458 mL
5 mM 0.4589 mL 2.2946 mL 4.5892 mL
10 mM 0.2295 mL 1.1473 mL 2.2946 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Wang P, et al. The Design and Synthesis of N-Xanthone Benzenesulfonamides as Novel Phosphoglycerate Mutase 1 (PGAM1) Inhibitors. Molecules. 2018 Jun 8;23(6). pii: E1396.

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