SU5205

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上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

SU5205  纯度: 98.44%

SU5205 是 VEGFR2 (FLK-1) 的抑制剂，IC50 值为 9.6 μM。

SU5205

SU5205 Chemical Structure

CAS No. : 3476-86-6

规格 价格 是否有货 数量
10 mM * 1 mL in DMSO ￥550 In-stock
50 mg ￥500 In-stock
100 mg ￥800 In-stock
200 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

SU5205 相关产品

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生物活性

SU5205 is an inhibitor of VEGFR2 (FLK-1), with an IC50 of 9.6 μM[1].

IC50 & Target[1]

Flk-1

9.6 μM (IC50)

体外研究
(In Vitro)

SU5205 inhibits ligand-induced endothelial mitogenesis for VEGF with an IC50 of 5.1 μM[1].

Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

239.24

Formula

C15H10FNO
CAS 号

3476-86-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
溶解性数据
In Vitro: 

DMSO : 250 mg/mL (1044.98 mM; Need ultrasonic)

配制储备液
浓度 溶剂体积 质量 1 mg 5 mg 10 mg
1 mM 4.1799 mL 20.8995 mL 41.7990 mL
5 mM 0.8360 mL 4.1799 mL 8.3598 mL
10 mM 0.4180 mL 2.0900 mL 4.1799 mL

*

请根据产品在不同溶剂中的溶解度选择合适的溶剂配制储备液；一旦配成溶液，请分装保存，避免反复冻融造成的产品失效。
储备液的保存方式和期限：-80°C, 6 months; -20°C, 1 month。-80°C 储存时，请在 6 个月内使用，-20°C 储存时，请在 1 个月内使用。
参考文献

  • [1]. Torsten K, et, al. Synthesis and radiopharmacological investigation of 3-[4′-[(18)F]fluorobenzylidene]indolin-2-one as possible tyrosine kinase inhibitor. Bioorg Med Chem. 2009 Nov 15; 17(22): 7732-42.

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