PKG inhibitor peptide TFA

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

PKG inhibitor peptide TFA 

PKG inhibitor peptide TFA 是一种 ATP 竞争性的 PKG 抑制剂，Ki 值为 86 μM。

PKG inhibitor peptide TFA

PKG inhibitor peptide TFA Chemical Structure

规格 是否有货
100 mg   询价  
250 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

PKG inhibitor peptide TFA 的其他形式现货产品:

PKG inhibitor peptide

生物活性

PKG inhibitor peptide TFA is an ATP-competitive inhibitor of cGMP-dependent protein kinase (PKG), with a Ki of 86 μM[1].

IC50 & Target

Ki: 86 μM (PKG)[1]
体外研究
(In Vitro)

Summary of experiments showing that intracellular dialysis of postsynaptic cells with PKG inhibitor PKG inhibitor peptide TFA (1 mM) failed to alter the induction of long-term depression (CCh-LTD)[2].

Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only.
分子量

1057.13

Formula

C40H75F3N18O12
Sequence

Arg-Lys-Arg-Ala-Arg-Lys-Glu
Sequence Shortening

RKRARKE
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Bhatnagar D, et al. Synthetic peptide analogues differentially alter the binding affinities of cyclic nucleotide dependent protein kinases for nucleotide substrates. Biochemistry. 1988 Mar 22;27(6):1988-94.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务