标签归档：aldha

ALDH1A3-IN-2

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-2 

ALDH1A3-IN-2 (Compound 15) 是一种有效的 ALDH1A3 抑制剂，IC50 为 0.30 μM。醛脱氢酶 (ALDH) 在包括前列腺癌在内的各种肿瘤类型中过度表达。ALDH1A3-IN-2 具有研究癌症疾病的潜力。

ALDH1A3-IN-2

ALDH1A3-IN-2 Chemical Structure

CAS No. : 886502-08-5

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250 mg   询价  
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生物活性

ALDH1A3-IN-2 (Compound 15) is a potent inhibitor of ALDH1A3 with an IC50 of 1.29 μM. Aldehyde dehydrogenases (ALDHs) are overexpressed in various tumor types including prostate cancer. ALDH1A3-IN-2 has the potential for the research of cancer diseases[1].

分子量

203.28

Formula

C13H17NO
CAS 号

886502-08-5
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ibrahim AIM, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH3A1-IN-2

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH3A1-IN-2 

ALDH3A1-IN-2 (Compound 19) 是一种有效的 ALDH3A1 抑制剂，IC50 为 1.29 μM。醛脱氢酶 (ALDH) 在包括前列腺癌在内的各种肿瘤类型中过度表达。ALDH3A1-IN-2 具有研究癌症疾病的潜力。

ALDH3A1-IN-2

ALDH3A1-IN-2 Chemical Structure

CAS No. : 374635-48-0

规格 是否有货
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250 mg   询价  
500 mg   询价  

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生物活性

ALDH3A1-IN-2 (Compound 19) is a potent inhibitor of ALDH3A1 with an IC50 of 1.29 μM. Aldehyde dehydrogenases (ALDHs) are overexpressed in various tumor types including prostate cancer. ALDH3A1-IN-2 has the potential for the research of cancer diseases[1].

分子量

222.24

Formula

C11H14N2O3
CAS 号

374635-48-0
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ibrahim AIM, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH3A1-IN-1

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH3A1-IN-1 

ALDH3A1-IN-1 (Compound 18) 是一种有效的 ALDH3A1 抑制剂，IC50 为 1.61 μM。ALDH3A1-IN-1 作为单药或与多西紫杉醇联合治疗，对患者来源的原发性前列腺肿瘤上皮细胞比 DEAB 更有效。

ALDH3A1-IN-1

ALDH3A1-IN-1 Chemical Structure

CAS No. : 1039855-56-5

规格 是否有货
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250 mg   询价  
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生物活性

ALDH3A1-IN-1 (Compound 18) is a potent inhibitor of ALDH3A1 with an IC50 of 1.61 μM. ALDH3A1-IN-1 is more potent than DEAB against patient-derived primary prostate tumor epithelial cells, as single agents or in combination treatment with docetaxel[1].

分子量

250.29

Formula

C13H18N2O3
CAS 号

1039855-56-5
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ibrahim AIM, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A1-IN-2

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A1-IN-2 

ALDH1A1-IN-2 是醛脱氢酶 1a1 (aldh1a1) 的有效抑制剂。醛脱氢酶 (ALDH) 构成酶家族，在氧化各种细胞毒性异种醛和生物醛中起关键作用。ALDH1A1-IN-2 具有研究癌症、炎症或肥胖症的潜力 (摘自专利 WO2019089626A1，化合物 295)。

ALDH1A1-IN-2

ALDH1A1-IN-2 Chemical Structure

CAS No. : 2231081-18-6

规格 价格 是否有货 数量
5 mg ￥3500 In-stock
10 mg ￥5600 In-stock
25 mg ￥11200 In-stock
50 mg   询价  
100 mg   询价  

* Please select Quantity before adding items.

ALDH1A1-IN-2 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Metabolism/Protease Compound Library
  • Anti-Cancer Compound Library
  • Glutamine Metabolism Compound Library
  • Anti-Cancer Metabolism Compound Library

生物活性

ALDH1A1-IN-2 is a potent inhibitor of aldehyde dehydrogenase 1a1 (aldh1a1). Aldehyde dehydrogenases (ALDH) constitute a family of enzymes that play a critical role in oxidizing various cytotoxic xenogenic and biogenic aldehydes. ALDH1A1-IN-2 has the potential for the research of cancer, inflammation, or obesity (extracted from patent WO2019089626A1, compound 295)[1].

分子量

494.99

Formula

C25H23ClN4O3S
CAS 号

2231081-18-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
参考文献

  • [1]. Shyh Ming YANG, et al. Substituted quinoline analogs as aldehyde dehydrogenase 1a1 (aldh1a1) inhibitors. Patent WO2019089626A1.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A1-IN-2

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A1-IN-2 

ALDH1A1-IN-2 是醛脱氢酶 1a1 (aldh1a1) 的有效抑制剂。醛脱氢酶 (ALDH) 构成酶家族，在氧化各种细胞毒性异种醛和生物醛中起关键作用。ALDH1A1-IN-2 具有研究癌症、炎症或肥胖症的潜力 (摘自专利 WO2019089626A1，化合物 295)。

ALDH1A1-IN-2

ALDH1A1-IN-2 Chemical Structure

CAS No. : 2231081-18-6

规格 价格 是否有货 数量
5 mg ￥3500 In-stock
10 mg ￥5600 In-stock
25 mg ￥11200 In-stock
50 mg   询价  
100 mg   询价  

* Please select Quantity before adding items.

ALDH1A1-IN-2 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Metabolism/Protease Compound Library
  • Anti-Cancer Compound Library
  • Glutamine Metabolism Compound Library
  • Anti-Cancer Metabolism Compound Library

生物活性

ALDH1A1-IN-2 is a potent inhibitor of aldehyde dehydrogenase 1a1 (aldh1a1). Aldehyde dehydrogenases (ALDH) constitute a family of enzymes that play a critical role in oxidizing various cytotoxic xenogenic and biogenic aldehydes. ALDH1A1-IN-2 has the potential for the research of cancer, inflammation, or obesity (extracted from patent WO2019089626A1, compound 295)[1].

分子量

494.99

Formula

C25H23ClN4O3S
CAS 号

2231081-18-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
参考文献

  • [1]. Shyh Ming YANG, et al. Substituted quinoline analogs as aldehyde dehydrogenase 1a1 (aldh1a1) inhibitors. Patent WO2019089626A1.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A1-IN-2

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A1-IN-2 

ALDH1A1-IN-2 是醛脱氢酶 1a1 (aldh1a1) 的有效抑制剂。醛脱氢酶 (ALDH) 构成酶家族，在氧化各种细胞毒性异种醛和生物醛中起关键作用。ALDH1A1-IN-2 具有研究癌症、炎症或肥胖症的潜力 (摘自专利 WO2019089626A1，化合物 295)。

ALDH1A1-IN-2

ALDH1A1-IN-2 Chemical Structure

CAS No. : 2231081-18-6

规格 价格 是否有货 数量
5 mg ￥3500 In-stock
10 mg ￥5600 In-stock
25 mg ￥11200 In-stock
50 mg   询价  
100 mg   询价  

* Please select Quantity before adding items.

ALDH1A1-IN-2 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Metabolism/Protease Compound Library
  • Anti-Cancer Compound Library
  • Glutamine Metabolism Compound Library
  • Anti-Cancer Metabolism Compound Library

生物活性

ALDH1A1-IN-2 is a potent inhibitor of aldehyde dehydrogenase 1a1 (aldh1a1). Aldehyde dehydrogenases (ALDH) constitute a family of enzymes that play a critical role in oxidizing various cytotoxic xenogenic and biogenic aldehydes. ALDH1A1-IN-2 has the potential for the research of cancer, inflammation, or obesity (extracted from patent WO2019089626A1, compound 295)[1].

分子量

494.99

Formula

C25H23ClN4O3S
CAS 号

2231081-18-6
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式
Powder -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
参考文献

  • [1]. Shyh Ming YANG, et al. Substituted quinoline analogs as aldehyde dehydrogenase 1a1 (aldh1a1) inhibitors. Patent WO2019089626A1.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A3-IN-1

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-1 

ALDH1A3-IN-1 (Compound 14) 是一个有效的 ALDH1A3 抑制剂，其 IC50 值为 0.63 µM，Ki 值为 0.46 µM。ALDH1A3-IN-1 能被用于研究前列腺癌 (prostate cancer)。

ALDH1A3-IN-1

ALDH1A3-IN-1 Chemical Structure

CAS No. : 1695970-90-1

规格 是否有货
100 mg   询价  
250 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

生物活性

ALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC50 of 0.63 µM and a Ki of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancer[1].

IC50 & Target

ALDH1A3

0.63 μM (IC50)

ALDH1A1

7.08 μM (IC50)

ALDH3A1

8.00 μM (IC50)

ALDH1A3

0.46 μM (Ki)

ALDH1A3

26.92 μM (Km)

体外研究
(In Vitro)

ALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate cancer cell lines[1].
ALDH1A3-IN-1 (0-200 µM, 72 h) reduces cell viability of primary prostate cells in a dose-dependent manner[1].

Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only.

Cell Proliferation Assay[1]

Cell Line: PC3, LNCaP, and DU145 cells
Concentration: 12.5-200 µM
Incubation Time: 96 h
Result: Showed antiproliferative activity with IC50 values of 47 ± 6, 25 ± 1, and 61 ± 5 µM against PC3, LNCaP, and DU145 cells.

Cell Viability Assay[1]

Cell Line: Primary cells cultured at early passage from human prostate tissue biopsies
Concentration: 50 and 200 μM
Incubation Time: 72 h
Result: Resulted a dose-dependent reduction in percentage cell viability of primary prostate epithelial cultures.

分子量

284.19

Formula

C13H18BrNO
CAS 号

1695970-90-1
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ali I M Ibrahim, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A3-IN-1

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-1 

ALDH1A3-IN-1 (Compound 14) 是一个有效的 ALDH1A3 抑制剂，其 IC50 值为 0.63 µM，Ki 值为 0.46 µM。ALDH1A3-IN-1 能被用于研究前列腺癌 (prostate cancer)。

ALDH1A3-IN-1

ALDH1A3-IN-1 Chemical Structure

CAS No. : 1695970-90-1

规格 是否有货
100 mg   询价  
250 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

生物活性

ALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC50 of 0.63 µM and a Ki of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancer[1].

IC50 & Target

ALDH1A3

0.63 μM (IC50)

ALDH1A1

7.08 μM (IC50)

ALDH3A1

8.00 μM (IC50)

ALDH1A3

0.46 μM (Ki)

ALDH1A3

26.92 μM (Km)

体外研究
(In Vitro)

ALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate cancer cell lines[1].
ALDH1A3-IN-1 (0-200 µM, 72 h) reduces cell viability of primary prostate cells in a dose-dependent manner[1].

上海金畔生物科技有限公司 has not independently confirmed the accuracy of these methods. They are for reference only.

Cell Proliferation Assay[1]

Cell Line: PC3, LNCaP, and DU145 cells
Concentration: 12.5-200 µM
Incubation Time: 96 h
Result: Showed antiproliferative activity with IC50 values of 47 ± 6, 25 ± 1, and 61 ± 5 µM against PC3, LNCaP, and DU145 cells.

Cell Viability Assay[1]

Cell Line: Primary cells cultured at early passage from human prostate tissue biopsies
Concentration: 50 and 200 μM
Incubation Time: 72 h
Result: Resulted a dose-dependent reduction in percentage cell viability of primary prostate epithelial cultures.

分子量

284.19

Formula

C13H18BrNO
CAS 号

1695970-90-1
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ali I M Ibrahim, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A3-IN-1

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-1 

ALDH1A3-IN-1 (Compound 14) 是一个有效的 ALDH1A3 抑制剂，其 IC50 值为 0.63 µM，Ki 值为 0.46 µM。ALDH1A3-IN-1 能被用于研究前列腺癌 (prostate cancer)。

ALDH1A3-IN-1

ALDH1A3-IN-1 Chemical Structure

CAS No. : 1695970-90-1

规格 是否有货
100 mg   询价  
250 mg   询价  
500 mg   询价  

* Please select Quantity before adding items.

生物活性

ALDH1A3-IN-1 (Compound 14) is a potent ALDH1A3 inhibitor, with an IC50 of 0.63 µM and a Ki of 0.46 µM. ALDH1A3-IN-1 can be studied in prostate cancer[1].

IC50 & Target

ALDH1A3

0.63 μM (IC50)

ALDH1A1

7.08 μM (IC50)

ALDH3A1

8.00 μM (IC50)

ALDH1A3

0.46 μM (Ki)

ALDH1A3

26.92 μM (Km)

体外研究
(In Vitro)

ALDH1A3-IN-1 (Compound 14) (0-200 µM, 96 h) shows antiproliferative activity in prostate cancer cell lines[1].
ALDH1A3-IN-1 (0-200 µM, 72 h) reduces cell viability of primary prostate cells in a dose-dependent manner[1].

Shanghai Jinpan Biotech Co Ltd has not independently confirmed the accuracy of these methods. They are for reference only.

Cell Proliferation Assay[1]

Cell Line: PC3, LNCaP, and DU145 cells
Concentration: 12.5-200 µM
Incubation Time: 96 h
Result: Showed antiproliferative activity with IC50 values of 47 ± 6, 25 ± 1, and 61 ± 5 µM against PC3, LNCaP, and DU145 cells.

Cell Viability Assay[1]

Cell Line: Primary cells cultured at early passage from human prostate tissue biopsies
Concentration: 50 and 200 μM
Incubation Time: 72 h
Result: Resulted a dose-dependent reduction in percentage cell viability of primary prostate epithelial cultures.

分子量

284.19

Formula

C13H18BrNO
CAS 号

1695970-90-1
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
参考文献

  • [1]. Ali I M Ibrahim, et al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A3-IN-3

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-3 

ALDH1A3-IN-3 (化合物 16) 是一种有效的 ALDH1A3 抑制剂，IC50 值为 0.26 μM。ALDH1A3-IN-3 也是 ALDH3A1 的底物。ALDH1A3-IN-3 可用于前列腺癌的研究。

ALDH1A3-IN-3

ALDH1A3-IN-3 Chemical Structure

CAS No. : 18962-05-5

规格 价格 是否有货 数量
1 g ￥350 In-stock
5 g   询价  
10 g   询价  

* Please select Quantity before adding items.

ALDH1A3-IN-3 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Fragment Library

生物活性

ALDH1A3-IN-3 (compound 16) is a potent inhibitor of ALDH1A3, with an IC50 of 0.26 μM. ALDH1A3-IN-3 is also a good ALDH3A1 substrate. ALDH1A3-IN-3 can be used for the research of prostate cancer[1].

IC50 & Target

IC50: 0.26 μM (ALDH1A3)[1]
分子量

164.20

Formula

C10H12O2
CAS 号

18962-05-5
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

4°C, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
参考文献

  • [1]. Ibrahim AIM, et, al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务

ALDH1A3-IN-3

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-3 

ALDH1A3-IN-3 (化合物 16) 是一种有效的 ALDH1A3 抑制剂，IC50 值为 0.26 μM。ALDH1A3-IN-3 也是 ALDH3A1 的底物。ALDH1A3-IN-3 可用于前列腺癌的研究。

ALDH1A3-IN-3

ALDH1A3-IN-3 Chemical Structure

CAS No. : 18962-05-5

规格 价格 是否有货 数量
1 g ￥350 In-stock
5 g   询价  
10 g   询价  

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ALDH1A3-IN-3 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Fragment Library

生物活性

ALDH1A3-IN-3 (compound 16) is a potent inhibitor of ALDH1A3, with an IC50 of 0.26 μM. ALDH1A3-IN-3 is also a good ALDH3A1 substrate. ALDH1A3-IN-3 can be used for the research of prostate cancer[1].

IC50 & Target

IC50: 0.26 μM (ALDH1A3)[1]
分子量

164.20

Formula

C10H12O2
CAS 号

18962-05-5
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

4°C, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
参考文献

  • [1]. Ibrahim AIM, et, al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

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ALDH1A3-IN-3

发表于由

上海金畔生物科技有限公司为生命科学和医药研发人员提供生物活性分子抑制剂、激动剂、特异性抑制剂、化合物库、重组蛋白，专注于信号通路和疾病研究领域。

ALDH1A3-IN-3 

ALDH1A3-IN-3 (化合物 16) 是一种有效的 ALDH1A3 抑制剂，IC50 值为 0.26 μM。ALDH1A3-IN-3 也是 ALDH3A1 的底物。ALDH1A3-IN-3 可用于前列腺癌的研究。

ALDH1A3-IN-3

ALDH1A3-IN-3 Chemical Structure

CAS No. : 18962-05-5

规格 价格 是否有货 数量
1 g ￥350 In-stock
5 g   询价  
10 g   询价  

* Please select Quantity before adding items.

ALDH1A3-IN-3 相关产品

•相关化合物库:

  • Bioactive Compound Library Plus
  • Fragment Library

生物活性

ALDH1A3-IN-3 (compound 16) is a potent inhibitor of ALDH1A3, with an IC50 of 0.26 μM. ALDH1A3-IN-3 is also a good ALDH3A1 substrate. ALDH1A3-IN-3 can be used for the research of prostate cancer[1].

IC50 & Target

IC50: 0.26 μM (ALDH1A3)[1]
分子量

164.20

Formula

C10H12O2
CAS 号

18962-05-5
运输条件

Room temperature in continental US; may vary elsewhere.
储存方式

4°C, stored under nitrogen

*In solvent : -80°C, 6 months; -20°C, 1 month (stored under nitrogen)
参考文献

  • [1]. Ibrahim AIM, et, al. Expansion of the 4-(Diethylamino)benzaldehyde Scaffold to Explore the Impact on Aldehyde Dehydrogenase Activity and Antiproliferative Activity in Prostate Cancer. J Med Chem. 2022 Mar 10;65(5):3833-3848.

所有产品仅用作科学研究或药证申报，我们不为任何个人用途提供产品和服务